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EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Rivista
Codice:
E060692
ISSN:
0223-5234
Dati Generali
Dati Generali
Pubblicazioni (63)
Pulisci
Ordina Pubblicazioni:
ascendente
decrescente
2-Substituted Benzothiazoles as Antiproliferative Agents: Novel Insights on Structure-Activity Relationships
Articolo
5-Arylisothiazol-3(2H)-one-1,(1)-(di)oxides: A new class of selective tumor-associated carbonic anhydrases (hCA IX and XII) inhibitors
Articolo
A novel life for antitumor combretastatins: Recent developments of hybrids, prodrugs, combination therapies, and antibody-drug conjugates
Articolo
A systematic review on the current status of PSMA-targeted imaging and radioligand therapy
Articolo
AMBER force field implementation of the boronate function to simulate the inhibition of beta-lactamases by alkyl and aryl boronic acids
Articolo
Anti-Candida activity and cytotoxicity of a large library of new N-substituted-1,3-thiazolidin-4-one derivatives
Articolo
Carvacrol prodrugs as novel antimicrobial agents
Articolo
Chalcogenides-incorporating carbonic anhydrase inhibitors concomitantly reverted oxaliplatin-induced neuropathy and enhanced antiproliferative action
Articolo
Chalcones: Unearthing their therapeutic possibility as monoamine oxidase B inhibitors
Articolo
Chemical Properties of Bile Acids. Part. 2. pKa Values in Water and Aqueous Methanol of Some Hydroxy Bile Acids
Articolo
Crystal structure of the Eg5 - K858 complex and implications for structure-based design of thiadiazole-containing inhibitors
Articolo
Cyclic tertiary sulfamates: selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
Articolo
Design, synthesis and biochemical evaluation of novel multi-target inhibitors as potential anti-Parkinson agents
Articolo
Design, synthesis and biological characterization of thiazolidin-4-one derivatives as promising inhibitors of Toxoplasma gondii
Articolo
Design, synthesis and biological evaluation of imidazole and triazole-based carbamates as novel aromatase inhibitors
Articolo
Design, synthesis, and biological activity of 2-aroylbenzofuran-3-ols and 2-aroylbenzofuran derivatives: A new route towards hMAO-B inhibition
Articolo
Development of benzene and benzothiazole-sulfonamide analogues as selective inhibitors of the tumor-associated carbonic anhydrase IX
Articolo
Development of glycine-α-methyl-proline-containing tripeptides with neuroprotective properties
Articolo
Development of linear β-turn inducers containing peptides as arc mimetics with DNA topological and sequence selectivity
Articolo
Discovery of 7-aminophenanthridin-6-one as a new scaffold for matrix metalloproteinase inhibitors with multitarget neuroprotective activity
Articolo
Discovery of gemfibrozil analogues that activate PPARa and enhance the expression of gene CPT1A involved in fatty acids catabolism
Articolo
Effect of milrinone analogues on intracellular calcium increase in single living H9C2 cardiac cells
Articolo
Effects of 3-(4’-geranyloxy-3’-methoxyphenyl)-2-trans propenoic acid and its ester derivatives on biofilm formation by two oral pathogens, Porphyromonas gingivalis and Streptococcus mutans
Articolo
Evaluation of a large library of (thiazol-2-yl)hydrazones and analogues as histone acetyltransferase inhibitors: enzyme and cellular studies
Articolo
Exploring 4-substituted-2-thiazolylhydrazones from 2-, 3-, and 4-acetylpyridine as selective and reversible hMAO-B inhibitors
Articolo
Extending pK(a) prediction accuracy: High-throughput pK(a) measurements to understand pK(a) modulation of new chemical series
Articolo
Fibrate-derived N-(methylsulfonyl)amides with antagonistic properties on PPARa
Articolo
Formation of micelles and liposomes from carnitine amphiphiles.
Articolo
Haloperidol metabolite II prodrug: Asymmetric synthesis and biological evaluation on rat C6 glioma cells
Articolo
Hybrid peptides endomorphin-2/DAMGO: Design, synthesis and biological evaluation
Articolo
Improving the solubility of a new class of antiinflammatory pharmacodynamic hybrids, that release nitric oxide and inhibit cycloxygenase-2 isoenzyme.
Articolo
In vitro and in vivo studies of gold(I) azolate/phosphane complexes for the treatment of basal like breast cancer
Articolo
Locally constrained xylene-based cyclic mimetics of SOCS3 protein
Articolo
Multitarget PPARγ agonists as innovative modulators of the metabolic syndrome
Articolo
New insights into the biological properties of Crocus sativus L.: chemical modifications, human monoamine oxidases inhibition and molecular modeling studies
Articolo
Novel 1,3-thiazolidin-4-one derivatives as promising anti-Candida agents endowed with anti-oxidant and chelating properties
Articolo
Novel anti-Alzheimer phenol-lipoyl hybrids: Synthesis, physico-chemical characterization, and biological evaluation
Articolo
Novel bisphosphonates with antiresorptive effect in bone mineralization and osteoclastogenesis
Articolo
O-derivatization of natural tropolone and β-thujaplicin leading to effective inhibitors of human carbonic anhydrases IX and XII
Articolo
Peptidyl 3-substituted 1-hydroxyureas as isosteric analogues of succinylhydroxamate MMP inhibitors
Articolo
Preparation of bivalent agonists for targeting the mu opioid and cannabinoid receptors
Articolo
Production, crystallographic studies, and functional profiling of γ-carbonic anhydrase from the probiotic Limosilactobacillus reuteri: In vitro and cell-based insights
Articolo
Recent advances in the development of selective human MAO-B inhibitors: (Hetero)arylidene-(4-substituted-thiazol-2-yl)hydrazines
Articolo
Resveratrol-based compounds and neurodegeneration: Recent insight in multitarget therapy
Articolo
Simplified analogues of ritanserin and their affinity at 5-HT2A, 5-HT2B and 5-HT2C serotonin receptors
Articolo
Structural development studies of PPARs ligands based on tyrosine scaffold
Articolo
Synthesis and activity of endomorphin-2 and morphiceptin analogues with proline surrogates in position 2
Articolo
Synthesis and anti-inflammatory effects of some bis(2-benzimidazolyl) thioethers and their copper(II) chelates orally administered in the rat.
Articolo
Synthesis and antiplatelet activity of thioaryloxyacids analogues of clofibric acid
Articolo
Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents
Articolo
Synthesis and cytotoxicity of novel (thiazol-2-yl) hydrazine derivatives as promising anti-Candida agents
Articolo
Synthesis and evaluation of new tripeptide phosphonate inhibitors of MMP-8 and MMP-2
Articolo
Synthesis and evalutation of 2-(5-methoxythiophen-3-yl)ethylamines as potential dopamine agonists
Articolo
Synthesis and in vitro selective anti-Helicobacter pylori activity of N-substituted-2-oxo-2H-1-benzopyran-3-carboxamides
Articolo
Synthesis and inhibitory activity against human monoamine oxidase of N1-thiocarbamoyl-3,5-di(hetero)aryl-4,5-dihydro-(1H)-pyrazole derivatives
Articolo
Synthesis and pharmacological screening of a large library of 1,3,4-thiadiazolines as innovative therapeutic tools for the treatment of prostate cancer and melanoma
Articolo
Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives
Articolo
Synthesis, anti-Candida activity, and cytotoxicity of new (4-(4-iodophenyl)thiazol-2-yl)hydrazine derivatives
Articolo
Synthesis, biological evaluation and quantitative structure-active relationships of 1,3-thiazolidin-4-one derivatives. A promising chemical scaffold endowed with high antifungal potency and low cytotoxicity
Articolo
Synthesis, biological evaluation, and docking study of indole aryl sulfonamides as aromatase inhibitors
Articolo
Synthesis, in vitro evaluation, and molecular modelling investigation of benzenesulfonimide Peroxisome Proliferator-Activated Receptors α antagonists
Articolo
Synthesis, structure-activity relationships and molecular docking studies of phenyldiazenyl sulfonamides as aromatase inhibitors
Articolo
Therapeutic potential for coxibs-nitric oxide releasing hybrids in cystic fibrosis.
Articolo
No Results Found
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